ZD0473 pharmacokinetics in Japanese patients: a Phase I dose-escalation study
References
- . Clinical pharmacokinetics and administration of established platinum drugs. Drugs. 2000;59(Suppl. 4):19–27
-
.
AMD473.
Drugs of the Future. 1998;23:1062–1065
- . Preclinical and clinical overview of the novel platinum complex, ZD0473 (cis-amminedichloro [2-methylpyridine] platinum [II]). Lung Cancer. 2000;29(Suppl. 1):70; (Abstr 227)
- . Activity of ZD0473 in small-cell lung cancer: an update in patients relapsing after one prior chemotherapy regimen. Eur J Cancer. 2001;37(Suppl. 6):S62; (Abstr 219)
-
.
Open-label Phase II study of ZD0473 in patients with metastatic hormone-refractory prostate cancer.
Eur Urol. 2002;1(Suppl. 1):158;
(Abstr 622)
- A Phase II trial of ZD0473 in patients with metastatic breast cancer. A National Cancer Institute of Canada Clinical Trials Group study (NCIC CTG-IND 129). Eur J Cancer. 2001;37(Suppl. 6):S194; (708)
- Pharmacokinetic (PK)/pharmacodynamic (PD) trial of the novel platinum compound ZD0473 administered as an iv infusion every 21 days. Eur J Cancer. 2001;37(Suppl. 6):S72; (Abstr 255)
- A validated liquid chromatography/tandem mass spectrometry assay for cis-amminedichloro-(2-methylpyridine)platinum(II) in human plasma ultrafiltrate. Anal Chem. 2002;74:591–599
-
Phase I and pharmacokinetic (PK) study of cis-amminedichloro(2-methylpyridine)platinum (II) (ZD0473), a novel sterically hindered platinum complex, in patients with metastatic hormone-refractory prostate cancer.
In:
Proc Am Soc Clin Oncol. 18:1999;p. 169;
(Abstr 648)
- . Clinical pharmacokinetics and dose optimisation of carboplatin. Clin Pharmacokinet. 1997;33:161–183
-
Oe T, Tian Y, O'Dwyer PJ, et al. Analysis of the platinum drug cis-amminedichloro(2-methylpyridine)platinum(II) in human urine by liquid chromatography/tandem mass spectrometry. J Chromatography (in press).
- ZD0473 phase II monotherapy trial in second-line non-small-cell lung cancer. Eur J Cancer. 2001;37(Suppl. 6):S59–S60 (Abstr 209)
- Pharmacokinetics of free and total platinum species after short-term infusion of cisplatin. Cancer Treat Rep. 1984;68:505–513
- . Carboplatin. A preliminary review of its pharmacodynamic and pharmacokinetic properties and therapeutic efficacy in the treatment of cancer. Drugs. 1989;37:162–190
PII: S0959-8049(02)80012-0
